Biological Activity Potent, non-substrate inhibitor of EAAT2 (GLT-1) that displays > 44-fold selectivity over EAAT1 and EAAT3 (IC50 values are 85, 3787 and 5004 nM for EAAT2, EAAT3 and EAAT1 respectively). Exhibits no activity towards ionotropic and metabotropic glutamate receptors.
Soluble to 100 mM in 1eq. NaOH and to 100 mM in DMSO
Desiccate at RT
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For batch specific data refer to the Certificate of Analysis.
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