6 results for "Casein Kinase 1 alpha Small Molecules and Peptides" in Products

Casein Kinase 1 alpha Small Molecules and Peptides

Casein kinases are a group of ubiquitous Ser/Thr kinases that phosphorylate key regulatory proteins involved in the control of cell differentiation, proliferation, chromosome segregation, circadian rhythms, and metabolic pathways. CK1 family members share a highly conserved kinase domain but differ in their variable N- and C-terminal domains. The C...

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CK1 inhibitor

Chemical Name: N-(2-Aminoethyl)-5-chloro-8-isoquinolinesulfonamide dihydrochloride
Purity: ≥99%
CK1 inhibitor
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Selective CK1 inhibitor. Also inhibits TGF-βRI

Chemical Name: 4-[4-(2,3-Dihydro-1,4-benzodioxin-6-yl)-5-(2-pyridinyl)-1H-imidazol-2-yl]benzamide
Purity: ≥98%
Selective CK1 inhibitor. Also inhibits TGF-βRI
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Potent CK1 inhibitor; also inhibits cyclin-dependent kinases

Chemical Name: 2-[[9-(1-Methylethyl)-6-[[3-(2-pyridinyl)phenyl]amino]-9H-purin-2-yl]amino]-1-butanol dihydrochloride
Purity: ≥98%
Potent CK1 inhibitor; also inhibits cyclin-dependent kinases
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Potent and selective CK1α, CK1δ and CK1ε inhibitor

Chemical Name: 4-(1-((4-Fluoro-1-methylpiperidin-4-yl)methyl)-4-(5-fluoropyridin-2-yl)-1H-imidazol-5-yl)-1H-pyrrolo[2,3-b]pyridine
Purity: ≥98%
Potent and selective CK1α, CK1δ and CK1ε inhibitor
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Cdk inhibitor; potently inhibits cdk1 and cdk2; also inhibits CK1; acts as molecular glue

Chemical Name: (2R)-2-[[9-(Methylethyl)-6-[[[4-(2-pyridinyl)phenyl]methyl]amino]-9H-purin-2-yl]amino]-1-butanol trihydrochloride
Purity: ≥98%
Cdk inhibitor; potently inhibits cdk1 and cdk2; also inhibits CK1; acts as molecular glue
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Potent and selective CK1α molecular glue Degrader

Chemical Name: 3-(5-(Benzo[d]isoxazol-3-ylamino)-1-oxoisoindolin-2-yl)piperidine-2,6-dione
Purity: ≥98%
Potent and selective CK1α molecular glue Degrader
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