4 results for "Group III mGluR Modulators" in Products

Group III mGluR Modulators

Potent mGlu5 antagonist; also positive allosteric modulator of mGlu4 receptors

Chemical Name: 2-Methyl-6-(phenylethynyl)pyridine hydrochloride
Purity: ≥98%
Potent mGlu5 antagonist; also positive allosteric modulator of mGlu4 receptors
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Selective positive allosteric modulator of group III mGlu receptors

Alternate Names: ML 396
Chemical Name: N-[3-Chloro-4-[(5-chloro-2-pyridinyl)oxy]phenyl]-2-pyridinecarboxamide
Purity: ≥98%
Selective positive allosteric modulator of group III mGlu receptors
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Positive allosteric modulator of mGlu7 and mGlu8 receptors; also NK1 antagonist; brain penetrant

Chemical Name: 3-(2,3-Difluoro-4-methoxyphenyl)-2,5-dimethyl-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidine
Purity: ≥98%
Positive allosteric modulators of mGlu7 and mGlu8 receptors; also NK1 antagonist; brain penetrant
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Negative allosteric modulator of mGlu7 receptors; brain penetrant

Chemical Name: 6-(2,4-Dimethylphenyl)-2-ethyl-6,7-dihydro-4(5H)-benzoxazolone
Purity: ≥98%
Negative allosteric modulator of mGlu7 receptors; brain penetrant
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