4 results for "TANK Binding Kinase Inhibitors Small Molecules and Peptides" in Products

TANK Binding Kinase Inhibitors Small Molecules and Peptides

TANK binding kinase (TBK) EC 2.7.11.1 is a ubiquitously expressed serine/threonine kinase belonging to the IκB Kinase (IKK) family, which regulates NF-κB signaling. This kinase has a range of substrates, leading to involvement in multiple pathways including immune response and inflammation, autophagy, cell proliferation and growth and insulin signaling.

TBK has a critical role in innate immunity and inflammation and functions downstream of multiple interferon (IFN) inducing pathways ...

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PDPK1 (PDK1) inhibitor

Chemical Name: N-[3-[[5-Iodo-4-[[3-[(2-thienylcarbonyl)amino]propyl]amino]-2-pyrimidinyl]amino]phenyl]-1-pyrrolidinecarboxamide
Purity: ≥98%
PDPK1 (PDK1) inhibitor
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Selective inhibitor of TBK

Chemical Name: 2-Amino-7-(1-methylethyl)-5-oxo-5H-[1]benzopyrano[2,3-b]pyridine-3-carboxylic acid
Purity: ≥98%
Selective inhibitor of TBK
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Potent TBK inhibitor

Chemical Name: N-[3-[[5-Cyclopropyl-2-[[4-(4-morpholinyl)phenyl]amino]-4-pyrimidinyl]amino]propyl]cyclobutanecarboxamide hydrochloride
Purity: ≥98%
Potent TBK inhibitor
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Salt inducible kinase (SIK) inhibitor; also ULK1 and 2 inhibitor

Chemical Name: N-[3-[[5-Cyclopropyl-2-[[3-(4-morpholinylmethyl)phenyl]amino]-4-pyrimidinyl]amino]propyl]cyclobutanecarboxamide dihydrochloride
Purity: ≥98%
Salt inducible kinase (SIK) inhibitor; also ULK1 and 2 inhibitor
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