CGP 7930

Catalog # Availability Size / Price Qty
1513/10
1513/50
CGP 7930 | CAS No. 57717-80-3 | GABA-B Receptor Modulators
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Description: Positive allosteric modulator of GABAB receptors

Chemical Name: 3,5-bis(1,1-Dimethylethyl)-4-hydroxy-β,β-dimethyl-benzenepropanol

Purity: ≥98%

Product Details
Citations (3)
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Biological Activity

Positive allosteric modulator of GABAB receptors. Increases the potency and efficacy of GABA at both native and recombinant GABAB receptors (EC50 values are 5.37 and 4.60μM respectively) and enhances the inhibitory effect of the agonist L-baclofen in cultured cortical neurons. Reduces operant self-administration of ethanol in alcohol-preferring rats following i.p. administration.

Technical Data

M.Wt:
292.46
Formula:
C19H32O2
Solubility:
Soluble to 100 mM in ethanol and to 100 mM in DMSO
Purity:
≥98%
Storage:
Desiccate at RT
CAS No:
57717-80-3

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
Tocris products are intended for laboratory research use only, unless stated otherwise.

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Citations for CGP 7930

The citations listed below are publications that use Tocris products. Selected citations for CGP 7930 include:

3 Citations: Showing 1 - 3

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