Biological Activitykisspeptin receptor (KISS1, GPR54) antagonist; kisspeptin-10 (Cat. No. 2570) analog. Inhibits kisspeptin-10 stimulation of inositol phosphate (IP) (IC50 = 7 nM) and release of gonadotrophin-releasing hormone (GnRH).
(Modifications: Ala-1 = D-Ala & N-terminal Ac, Trp-8 = D-Trp, Phe-10 = C-terminal amide)
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For batch specific data refer to the Certificate of Analysis.
Tocris products are intended for laboratory research use only, unless stated otherwise.
Discovery of potent kisspeptin antagonists delineate physiological mechanisms of gonadototrophin regulation.
Roseweir et al.
Citations for Kisspeptin 234
The citations listed below are publications that use Tocris products. Selected citations for Kisspeptin 234 include:
2 Citations: Showing 1 - 2
The pregnant mouse uterus exhibits a functional kisspeptin/KISS1R signaling system on the day of embryo implantation.
Authors: Fayazi Et al.
Am J Physiol Renal Physiol 2015;13:105
GPR54-dependent stimulation of luteinizing hormone secretion by neurokinin B in prepubertal rats.
Authors: Grachev Et al.
Reprod Biol Endocrinol 2012;7:e44344
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