Having trouble trying to find the right product? Chat with our scientists below - we're here to help!
5 results for "CHRM4" in Products
CHRM4 Products
Muscarinic acetylcholine receptor M4 is an Acetylcholine Receptor. Unlike muscarinic receptor M2, the M4 receptor is not involved in smooth muscle contraction. The clinical relevance of this receptor is unknown. However, mouse studies have linked it to adenylyl cyclase inhibition. Muscarinic acetylcholine receptor M4 has been reported to be expressed in many regions of the rat brain, particularly the striatum and hippocampus. ESTs have been isolated from human breast and eye libraries.
Selective M2 antagonist
| Alternate Names: | Otenzepad |
| Chemical Name: | 11-[[2-[(Diethylamino)methyl]-1-piperidinyl]acetyl]-5,11-dihydro-6H-pyrido[2,3-b][1,4]benzodiazepin-6-one |
| Purity: | ≥98% |
Loading...
Potent M2/M4 antagonist
| Chemical Name: | N-[2-[2-[(Dipropylamino)methyl]-1-piperidinyl]ethyl]-5,6-dihydro-6-oxo-11H-pyrido[2,3-b][1,4]benzodiazepine-11-carboxamide |
| Purity: | ≥98% |
Loading...
High affinity and selective M2 antagonist
| Chemical Name: | 11-[[4-[4-(Diethylamino)butyl]-1-piperidinyl]acetyl]-5,11-dihydro-6H-pyrido[2,3-b][1,4]benzodiazepin-6-one |
| Purity: | ≥98% |
Loading...
Selective M4 antagonist
| Chemical Name: | 3,6a,11,14-Tetrahydro-9-methoxy-2-methyl-(12H)-isoquino[1,2-b]pyrrolo[3,2-f][1,3]benzoxazine-1-carboxylic acid, ethyl ester |
| Purity: | ≥98% |
Loading...
Potent and selective M4 mAChR antagonist
| Chemical Name: | (3aR,5s,6aS)-2-((Tetrahydro-2H-pyran-4-yl)methyl)-N-(6-(2,3,5-trifluorophenyl)pyridazin-3-yl)octahydrocyclopenta[c]pyrrol-5-amine hydrochloride |
| Purity: | ≥98% |
Loading...