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3 results for "GPER/GPR30" in Products
GPER/GPR30 Products
GPR30 a former orphan receptor has been linked to estrogen-mediated activation of adenylyl cyclase, release of epidermal growth factor (EGF)-related ligands, and specific estrogen binding.1 GPR30 acts independently of estrogen receptors, ERalpha and ERbeta, to release of heparin-binding EGF and may play a role in breast cancer tumorogenesis.
High affinity and selective GPER antagonist
| Chemical Name: | (3aS*,4R*,9bR*)-4-(6-Bromo-1,3-benzodioxol-5-yl)-3a,4,5,9b-3H-cyclopenta[c]quinoline |
| Purity: | ≥98% |
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Selective GPER antagonist
| Chemical Name: | (±)-(3aR*,4S*,9bS*)-4-(6-Bromo-1,3-benzodioxol-5-yl)-3a,4,5,9b-tetrahydro-8-(1-methylethyl)-3H-cyclopenta[c]quinoline |
| Purity: | ≥98% |
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Potent and selective G protein-coupled estrogen receptor (GPER) antagonist
| Chemical Name: | N-[2-Cyclohexyl-4-(1-methylethyl)phenyl]-4-methoxybenzenemethanamine hydrochloride |
| Purity: | ≥98% |
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