18 results for "Additional Transcription Factor Compounds" in 产品

Additional Transcription Factor Compounds

Core binding factor inhibitor; attenuates hematopoiesis

Alternate Names: CBF&#946-Runx1 inhibitor II
Chemical Name: 7-Chloro-1,3-dihydro-5-(1H-pyrrol-2-yl)-2H-1,4-benzodiazepin-2-one
Purity: ≥98%
Core binding factor inhibitor; attenuates hematopoiesis
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YAP inhibitor

Alternate Names: Visudyne
Chemical Name: (4R,4aS)-18-Ethenyl-4,4a-dihydro-3,4-bis(methoxycarbonyl)-4a,8,14,19-tetramethyl-24H,26H-benzo[b]porphine-9,13-dipropanoic acid monomethyl ester
Purity: ≥95%
YAP inhibitor
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Selective Smad3 inhibitor; inhibits TGF-βR1 signaling

Chemical Name: 1,2,3,4-Tetrahydro-6,7-dimethoxy-2-[(2E)-3-(1-phenyl-1H-pyrrolo[2,3-b]pyridin-3-yl)-1-oxo-2-propenyl]-isoquinoline hydrochloride
Purity: ≥97%
Selective Smad3 inhibitor; inhibits TGF-βR1 signaling
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Potent and selective Foxo1 inhibitor; orally bioavailable

Chemical Name: 5-Amino-7-(cyclohexylamino)-1-ethyl-6-fluoro-1,4-dihydro-4-oxo-3-quinolinecarboxylic acid
Purity: ≥98%
Potent and selective Foxo1 inhibitor; orally bioavailable
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Hepatocyte nuclear factor 4α (HNF4α) antagonist

Chemical Name: 2-Methyl-1-[(2-methyl-5-nitrophenyl)sulfonyl]-1H-benzimidazole
Purity: ≥98%
Hepatocyte nuclear factor 4α (HNF4α) antagonist
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Brachyury down modulator

Chemical Name: (E)-4-(Dimethylamino)-N-[1-[4-fluoro-3-(2,2,2-trifluoroethoxy)anilino]-6-methoxy-7-isoquinolyl]but-2-enamide
Purity: ≥98%
Brachyury down modulator
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Potent and selective CREB inhibitor

Chemical Name: 3-(3-Aminopropoxy)-N-[2-[[3-[[(4-chloro-2-hydroxyphenyl)amino]carbonyl]-2-naphthalenyl]oxy]ethyl]-2-naphthalenecarboxamide hydrochloride
Purity: ≥98%
Potent and selective CREB inhibitor
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Steroid receptor coactivator 3 (SRC-3) inhibitor

Chemical Name: 1-(2-Pyridinyl)ethanone 2-(1-methyl-1H-benzimidazol-2-yl)hydrazone hydrochloride
Purity: ≥98%
Steroid receptor coactivator 3 (SRC-3) inhibitor
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Cryptochrome protein stabilizer; lengthens circadian period

Chemical Name: N-[3-(9H-Carbazol-9-yl)-2-hydroxypropyl]-N-(2-furanylmethyl)methanesulfonamide
Purity: ≥98%
Cryptochrome protein stabilizer; lengthens circadian period
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GLI antagonist; inhibits Hedgehog (Hh) signaling

Chemical Name: 2,2'-[[Dihydro-2-(4-pyridinyl)-1,3(2H,4H)-pyrimidinediyl]bis(methylene)]bis[N,N-dimethylbenzenamine
Purity: ≥98%
GLI antagonist; inhibits Hedgehog (Hh) signaling
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TRIM24 Degrader (PROTAC®)

Chemical Name: (2S,4R)-1-((S)-15-(tert-Butyl)-1-(3-(N-(1,3-dimethyl-2-oxo-6-(3-propoxyphenoxy)-2,3-dihydro-1H-benzo[d]imidazol-5-yl)sulfamoyl)phenyl)-1,13-dioxo-5,8,11-trioxa-2,14-diazahexadecan-16-oyl)-4-hydroxy-N-(4-(4-methylthiazol-5-yl)benzyl)pyrrolidine-2-carboxamide
Purity: ≥98%
TRIM24 Degrader (PROTAC®)
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Potent and reversible inhibitor of TEAD mediated Hippo/Yap signalling

Chemical Name: 4-[3-(2-Cyclohexylethoxy)benzoyl]-N-phenyl-1-piperazinecarboxamide
Purity: ≥98%
Potent and reversible inhibitor of TEAD mediated Hippo/Yap signalling
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Potent pan-TEAD inhibitor

Chemical Name: N-[(1S)-1-(2-Pyridinyl)ethyl]-5-[4-(trifluoromethyl)phenyl]-2-naphthalenecarboxamide
Purity: ≥98%
Potent pan-TEAD inhibitor
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High affinity Myc inhibitor

Chemical Name: 4-[2-(2-Furanyl)-6-(4-nitrophenyl)-4-pyridinyl]benzamide
Purity: ≥98%
High affinity Myc inhibitor
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Inhibits c-Myc-Max dimerization

Chemical Name: 5-[(4-Ethylphenyl)methylene]-2-thioxo-4-thiazolidinone
Purity: ≥98%
Inhibits c-Myc-Max dimerization
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High affinity Nur77 agonist

Chemical Name: Ethyl 3,5-dihydroxy-2-(1-oxooctyl)-benzeneacetate
Purity: ≥98%
High affinity Nur77 agonist
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Selective inhibitor of ATF6α; sensitizes cells to ER stress

Chemical Name: N-[1-[[2,4-bis(Trifluoromethyl)phenyl]methyl]-1H-pyrazol-4-yl]-5-(2-furanyl)-3-isoxazolecarboxamide
Purity: ≥98%
Selective inhibitor of ATF6α; sensitizes cells to ER stress
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YAP inhibitor

Purity: ≥95%
Peptide inhibitor of YAP signaling
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