Atovaquone

Catalog #: 6358 Datasheet / COA / SDS

Discontinued Product

6358 has been discontinued.
View all Oxidative Phosphorylation Inhibitors products.
Atovaquone | CAS No. 95233-18-4 | Oxidative Phosphorylation Inhibitors
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Description: Inhibits complex III of mitochondrial electron transport chain in parasites

Chemical Name: 2-[trans-4-(4-Chlorophenyl)cyclohexyl]-3-hydroxy-1,4-naphthalenedione

Purity: ≥98%

Product Details
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Biological Activity

Broad spectrum antiparasitic and antipneumocystic compound. Inhibits bc1 complex (complex III) of mitochondrial electron transport chain (EC50 = 0.26 μM), causing cell death in Plasmodium yoelii infected erythrocytes. Also inhibits DHODH. Also exhibits anti-MERS-CoV activity in Vero cells in vitro (IC50 = 0.72 μM).

Technical Data

M.Wt:
366.84
Formula:
C22H19ClO3
Solubility:
Soluble to 20 mM in DMSO
Purity:
≥98%
Storage:
Store at -20°C
CAS No:
95233-18-4

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
Tocris products are intended for laboratory research use only, unless stated otherwise.

Background References

  1. Efficacy of a hydroxynaphthoquinone, 566C80, in experimental Pneumocystis carinii pneumonitis.
    Hughes et al.
    Antimicrob.Agents Chemother., 1990;34:225
  2. Atovaquone, a broad spectrum antiparasitic drug, collapses mitochondrial membrane potential in a malarial parasite.
    Srivastava et al.
    J.Biol.Chem., 1997;272:3961
  3. Screening of FDA-approved drugs using a MERS-CoV clinical isolate from South Korea identifies potential therapeutic options for COVID-19.
    Ko et al.
    BioRxiv - Paper not yet peer reviewed, 2020;

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