BAN ORL 24

  ( 1 citations )    
Product Datasheet
Catalog Number:3661
Chemical Name:(2R)-1-(Phenylmethyl)-N-[3-(spiro[isobenzofuran-1(3H),4'-piperidin]-1-yl)propyl-2-pyrrolidinecarboxamide
Product Details
Citations (1)
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Biological Activity
Potent and selective NOP receptor antagonist (IC50 values are 0.27, 2500, 6700 and > 10000 nM for NOP, κ-, μ- and δ-receptors respectively). Inhibits nociceptin-induced stimulation of [35S]-GTPγS binding and Ca2+ mobilization in CHO cells in vitro and antagonizes NOP agonist-induced reduction in locomotor activity in vivo. Brain penetrant.
Technical Data
  • M.Wt:
    506.51
  • Formula:
    C27H35N3O2.2HCl
  • Solubility:
    Soluble to 100 mM in water and to 100 mM in DMSO
  • Purity:
    >97
  • Storage:
    Store at -20°C
  • CAS No:
    1401463-54-4
The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis. All Tocris products are intended for laboratory research use only.
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Citations:

The citations listed below are publications that use Tocris products. Selected citations for BAN ORL 24 include:

1 Citations: Showing 1 - 1

  1. Metformin induces PGC-1α expression and selectively affects hepatic PGC-1α functions.
    Authors: Aatsinki Et al.
    Am J Physiol Cell Physiol  2014;171:2351

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