Cysteinyl leukotriene receptor antagonist with equal affinity at both CysLT1
values are 6.8 and 6.5 respectively). Competitive antagonist of LTC4
- and LTE4
-induced contractions of the guinea pig trachea.
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Cysteinyl leukotriene receptors in the human lung: what's new?
Goranne et al.
Functional characteristics of cysteinyl-leukotriene receptor subtypes.
Life Sci., 2002;71:611
A second cysteinyl leukotriene receptor in human lung.
Labat et al.