Catalog Number: 2842
Biological Activity
Somatostatin sst5 receptor agonist (Ki values are 7.3, 13.5, 31.3 and 141 nM for sst5, sst2, sst1 and sst4 receptors respectively). Stimulates gastric emptying following i.c. administration.
Technical Data
  • M.Wt:
    1122.3
  • Formula:
    C61H75N11O10
  • Sequence:
    FFFWKTFT

    (Modifications: Phe-1 = D-Phe, Trp-4 = D-Trp, Thr-8 = C-terminal amide)

  • Solubility:
    Soluble to 1 mg/ml in water
  • Storage:
    Store at -20°C
  • CAS No:
    133073-82-2
The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis. All Tocris products are intended for laboratory research use only.
Background References
  1. Intracisternal injection of somatostatin receptor 5-preferring agonists induces a vagal cholinergic stimulation of gastric emptying in rats.
    Martinez et al.
    J.Pharmacol.Exp.Ther., 2000;293:1099
  2. Pharmacological characterisation of the goldfish somatostatin sst5 receptor.
    Nunn et al.
    Eur.J.Pharmacol., 2002;436:173
  3. Subtype selectivity of peptide analogs for all five cloned human somatostatin receptors (hsstr 1-5).
    Patel and Srikant
    Endocrinology, 1994;135:2814

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