(±)-Bisoprolol hemifumarate

  ( 3 citations )    
Product Datasheet
Catalog Number:0914
Chemical Name:(±)-1-[4-[[2-(1-Methylethoxy)ethoxy)methyl]phenoxy]-3-[(1-methylethyl)amino]-2-propanol hemifumarate
Product Details
Citations (3)
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Reviews
Biological Activity
A selective β1-adrenergic antagonist. Has a Kd of 2-3 nM at the β1 receptor and a β1/β2 selectivity of approximately 100-fold.
Technical Data
  • M.Wt:
    383.48
  • Formula:
    C18H31NO4.½C4H4O4
  • Solubility:
    Soluble to 50 mM in water
  • Purity:
    >98
  • Storage:
    Store at RT
  • CAS No:
    104344-23-2
The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis. All Tocris products are intended for laboratory research use only.
Product Datasheets
Citations:

The citations listed below are publications that use Tocris products. Selected citations for (±)-Bisoprolol hemifumarate include:

3 Citations: Showing 1 - 3
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  1. Recruitment of β-arrestin 1 and 2 to the β2-adrenoceptor: analysis of 65 ligands.
    Authors: Littmann Et al.
    PLoS One  2015;355:183
  2. Predicting in vivo cardiovascular properties of β-blockers from cellular assays: a quantitative comparison of cellular and cardiovascular pharmacological responses.
    Authors: Baker Et al.
    FASEB J  2011;25:4486
  3. Increased PKA activity and its influence on isoprenaline-stimulated L-type Ca2+ channels in the heart from ovariectomized rats.
    Authors: Kam Et al.
    Br J Pharmacol  2005;144:972

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