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(±)-Bisoprolol hemifumarate

0914 3 Citations Datasheet / COA / SDS
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(±)-Bisoprolol hemifumarate | CAS No. 104344-23-2 | Adrenergic beta-1 Receptor Antagonists
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Description: β1 antagonist

Chemical Name: (±)-1-[4-[[2-(1-Methylethoxy)ethoxy)methyl]phenoxy]-3-[(1-methylethyl)amino]-2-propanol hemifumarate

Purity: ≥98%

Product Details
Citations (3)
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Biological Activity

A selective β1-adrenergic antagonist. Has a Kd of 2-3 nM at the β1 receptor and a β1/β2 selectivity of approximately 100-fold.

Technical Data

M.Wt:
383.48
Formula:
C18H31NO4.½C4H4O4
Solubility:
Soluble to 50 mM in water
Purity:
≥98%
Storage:
Store at RT
CAS No:
104344-23-2

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
Tocris products are intended for laboratory research use only, unless stated otherwise.

Product Datasheets

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Citations for (±)-Bisoprolol hemifumarate

The citations listed below are publications that use Tocris products. Selected citations for (±)-Bisoprolol hemifumarate include:

3 Citations: Showing 1 - 3

  1. Recruitment of β-arrestin 1 and 2 to the β2-adrenoceptor: analysis of 65 ligands.
    Authors: Littmann Et al.
    PLoS One  2015;355:183
  2. Predicting in vivo cardiovascular properties of β-blockers from cellular assays: a quantitative comparison of cellular and cardiovascular pharmacological responses.
    Authors: Baker Et al.
    FASEB J  2011;25:4486
  3. Increased PKA activity and its influence on isoprenaline-stimulated L-type Ca2+ channels in the heart from ovariectomized rats.
    Authors: Kam Et al.
    Br J Pharmacol  2005;144:972

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VersaClone cDNA Plasmids

Human ADRB1 (P08588) VersaClone cDNA

RDC0259

Human beta-1 Adrenergic R/ADRB1 (NP_000675) VersaClone cDNA

RDC0630

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