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(±)-Bisoprolol hemifumarate

  ( 3 citations )    
Product Datasheet
Catalog Number:0914
Chemical Name:(±)-1-[4-[[2-(1-Methylethoxy)ethoxy)methyl]phenoxy]-3-[(1-methylethyl)amino]-2-propanol hemifumarate
Product Details
Citations (3)
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Reviews
Biological Activity
A selective β1-adrenergic antagonist. Has a Kd of 2-3 nM at the β1 receptor and a β1/β2 selectivity of approximately 100-fold.
Technical Data
  • M.Wt:
    383.48
  • Formula:
    C18H31NO4.½C4H4O4
  • Solubility:
    Soluble to 50 mM in water
  • Purity:
    >98
  • Storage:
    Store at RT
  • CAS No:
    104344-23-2
The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis. All Tocris products are intended for laboratory research use only.
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Citations:

The citations listed below are publications that use Tocris products. Selected citations for (±)-Bisoprolol hemifumarate include:

3 Citations: Showing 1 - 3
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  1. Recruitment of β-arrestin 1 and 2 to the β2-adrenoceptor: analysis of 65 ligands.
    Authors: Littmann Et al.
    PLoS One  2015;355:183
  2. Predicting in vivo cardiovascular properties of β-blockers from cellular assays: a quantitative comparison of cellular and cardiovascular pharmacological responses.
    Authors: Baker Et al.
    FASEB J  2011;25:4486
  3. Increased PKA activity and its influence on isoprenaline-stimulated L-type Ca2+ channels in the heart from ovariectomized rats.
    Authors: Kam Et al.
    Br J Pharmacol  2005;144:972

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