Chemical Name: (2E)-2-(1,3-Benzothiazol-2-yl)-3-[9-methyl-2-(3-methylphenoxy)-4-oxo-4H-pyrido[1,2-a]pyrimidin-3-yl]acrylonitrile
Biological ActivityCCG 63802 is a reversible inhibitor of regulator of G-protein signaling (RGS) proteins. Selective amongst RGS proteins, with greatest potency at RGS4. Inhibits GTPase accelerating protein activity of RGS4 and blocks its interaction with Gαo. Retains activity under reducing conditions.
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Tocris products are intended for laboratory research use only, unless stated otherwise.
Reversible, allosteric small-molecule inhibitors of regulator of G protein signaling proteins.
Blazer et al.
Citation for CCG 63802
The citations listed below are publications that use Tocris products. Selected citations for CCG 63802 include:
1 Citation: Showing 1 - 1
A new model of nerve injury in the rat reveals a role of Regulator of G protein Signaling 4 in tactile hypersensitivity.
Authors: Taccola Et al.
Experimental Neurology 2016;286:1
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