Reversible inhibitor of regulator of G-protein signaling (RGS) proteins. Selective amongst RGS proteins, with greatest potency at RGS4. Inhibits GTPase accelerating protein activity of RGS4 and blocks its interaction with Gαo
. Retains activity under reducing conditions.
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Reversible, allosteric small-molecule inhibitors of regulator of G protein signaling proteins.
Blazer et al.
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