CCG 63802

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4028/10
4028/50
CCG 63802 | CAS No. 620112-78-9 | Regulators of G Protein Signaling (RGS) Inhibitors
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Description: Inhibitor of regulator of G-protein signaling 4 (RGS4) protein

Chemical Name: (2E)-2-(1,3-Benzothiazol-2-yl)-3-[9-methyl-2-(3-methylphenoxy)-4-oxo-4H-pyrido[1,2-a]pyrimidin-3-yl]acrylonitrile

Purity: ≥99%

Product Details
Citations (1)
Reviews

Biological Activity

Reversible inhibitor of regulator of G-protein signaling (RGS) proteins. Selective amongst RGS proteins, with greatest potency at RGS4. Inhibits GTPase accelerating protein activity of RGS4 and blocks its interaction with Gαo. Retains activity under reducing conditions.

Technical Data

M.Wt:
450.51
Formula:
C26H18N4O2S
Solubility:
Soluble to 5 mM in DMSO with gentle warming
Purity:
≥99%
Storage:
Store at +4°C
CAS No:
620112-78-9

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
Tocris products are intended for laboratory research use only, unless stated otherwise.

Background References

  1. Reversible, allosteric small-molecule inhibitors of regulator of G protein signaling proteins.
    Blazer et al.
    Mol.Pharmacol., 2010;78:524

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Citation for CCG 63802

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