Catalog Number: 3500
Chemical Name: rel-5-(1,1-Dimethylheptyl)-2-[(1R,3S)-3-hydroxycyclohexyl]phenol
Biological Activity
Potent CB1 receptor agonist (Ki = 2.2 nM). Exhibits analgesic, motor depressant, anticonvulsant and hypothermic effects in vivo.
Technical Data
  • M.Wt:
    318.49
  • Formula:
    C21H34O2
  • Solubility:
    Soluble to 100 mM in DMSO and to 100 mM in ethanol
  • Purity:
    >98%
  • Storage:
    Store at -20°C
  • CAS No:
    70434-82-1
The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis. All Tocris products are intended for laboratory research use only.
Background References
  1. Cannabimimetic activity from CP-47,497, a derivative of 3-phenylcyclohexanol.
    Weissman et al.
    J.Pharmacol.Exp.Ther., 1982;223:516
  2. Structure-activity relationships for cannabinoid receptor-binding and analgesic activity: studies of bicyclic cannabinoid analogs.
    Melvin et al.
    Mol.Pharmacol., 1993;44:1008
  3. Synthesis and pharmacology of 1-deoxy analogs of CP-47,497 and CP-55,940.
    Huffman et al.
    Bioorg.Med.Chem., 2008;16:322

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