DPCPX

Tocris Bioscience | Catalog # 0439

Selective A1 antagonist
Tocris Bioscience

Key Product Details

Description

Selective A1 antagonist
View all Adenosine A1 Receptor Antagonists »

Product Description

DPCPX is a potent and selective A1 adenosine receptor antagonist, both in vitro and in vivo. Ki values are 3.9, 130, 50 and 4000 nM for human A1, A2A, A2B and A3 receptors respectively.

Product Specifications for DPCPX

Molecular Weight

304.39

Formula

C16H24N4O2

Storage

Store at RT

Purity

≥98% (HPLC)

Chemical Name

8-Cyclopentyl-1,3-dipropylxanthine

CAS Number

102146-07-6

PubChem ID

1329

InChI Key

FFBDFADSZUINTG-UHFFFAOYSA-N

SMILES

CCCN1C2=C(N=C(N2)C2CCCC2)C(=O)N(CCC)C1=O

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.

Solubility

Solvent Max Conc. mg/mL Max Conc. mM
Solubility
DMSO 1.52 5 with gentle warming
Ethanol 3.04 10 with gentle warming

Preparing Stock Solutions for DPCPX

The following data is based on the product molecular weight 304.39.

Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which all affect the solvent volumes required to prepare stock solutions.

Select a batch to recalculate based on the batch molecular weight:

Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 32.85 mL 164.26 mL 328.53 mL
0.5 mM 6.57 mL 32.85 mL 65.71 mL
1 mM 3.29 mL 16.43 mL 32.85 mL
5 mM 0.66 mL 3.29 mL 6.57 mL

Calculators

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Background References

References are publications that support the biological activity of the product. See our Citations tab to view 301 publications citing the usage of this product.

Product Documents for DPCPX

Certificate of Analysis

To download a Certificate of Analysis, please enter a lot or batch number in the search box below.

Product Specific Notices for DPCPX

For research use only

Customer Reviews for DPCPX (1)

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  • A selective A1 receptor antagonist
    Name: Anonymous
    Species: Rat
    Assay Type: Ex Vivo
    Verified Customer | Posted 02/06/2018
    This a selective A1 receptor antagonist. We used at 100nM in rat brain slice.

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