Potent and selective μ
-opioid receptor agonist (Ki
values are 7.0, 151 and 470 nM for μ
- and κ
-opioid receptors respectively). Displays antinociceptive activity in vivo
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All Tocris products are intended for laboratory research use only.
Receptor reserve and affinity of mu-opioid agonists in mouse antinociception: correlation with receptor binding.
Zernig et al.
Life Sci., 1995;57:2113
Opioid activity of C8813, a novel and potent opioid analgesic.
Liu et al.
Life Sci., 2003;73:233
Opioid interactions in rhesus monkeys: effects of δ + μ and δ + κ agonists on schedule-controlled responding and thermal nociception.
Stevenson et al.