Catalog Number: 3247
Alternate Names: Phentanyl citrate
Chemical Name: N-Phenyl-N-[1-(2-phenylethyl)-4-piperidinyl]propanamide citrate
Biological Activity
Potent and selective μ-opioid receptor agonist (Ki values are 7.0, 151 and 470 nM for μ-, δ- and κ-opioid receptors respectively). Displays antinociceptive activity in vivo.
Technical Data
  • M.Wt:
    528.59
  • Formula:
    C22H28N2O.C6H8O7
  • Solubility:
    Soluble to 40 mM in water
  • Purity:
    >99%
  • Storage:
    Store at RT
  • CAS No:
    990-73-8
The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis. All Tocris products are intended for laboratory research use only.
Background References
  1. Receptor reserve and affinity of mu-opioid agonists in mouse antinociception: correlation with receptor binding.
    Zernig et al.
    Life Sci., 1995;57:2113
  2. Opioid activity of C8813, a novel and potent opioid analgesic.
    Liu et al.
    Life Sci., 2003;73:233
  3. Opioid interactions in rhesus monkeys: effects of δ + μ and δ + κ agonists on schedule-controlled responding and thermal nociception.
    Stevenson et al.
    J.Pharmacol.Exp.Ther., 2003;307:1054

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