A very potent and selective inhibitor of dopamine uptake (IC50
for inhibition of [3
H]-dopamine uptake in rat striatal synaptosomes is 1.8 nM).
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All Tocris products are intended for laboratory research use only.
GBR 12783, a potent and selective inhibitor of dopamine uptake: biochemical studies in vivo and ex vivo.
Bonnet and Constentin
Cloning, pharmacological characterization and chromosome assignment of the human dopamine transporter.
Giros et al.
Evidence for the sequential formation of two complexes between an uptake inhibitor, GBR 12783 [1-[2-(diphenylmethoxy)ethyl]-4-(3-phenyl-2-propenyl)piperazine], and the neuronal transporter of dopamine.
Do-Rego et al.
In vivo labelling of the neuronal dopamine uptake complex in the mouse striatum by [3H]GBR 12783.
Vaugeois et al.
The citations listed below are publications that use Tocris products. Selected citations for GBR 12783 dihydrochloride include:
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