Binds with high affinity to MT3
melatonin sites in hamster brain, and low affinity (and no efficacy) at MT1
melatonin receptors and thus can be used to discriminate between the melatonin receptor subtypes.
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All Tocris products are intended for laboratory research use only.
Melatonin receptors: are there multiple subtypes?
Investigation into the contractile response of melatonin in the guinea-pig isolated proximal colon: the role of 5-HT4 and melatonin receptors.
Lucchelli et al.
The citations listed below are publications that use Tocris products. Selected citations for GR 135531 include:
Showing Results 1 - 5 of 5