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Catalog Number:2419
Chemical Name:5-Cyclohexyl-1-[4-(1H-imidazol-5-yl)-1-piperidinyl]-1-pentanone
Product Details
Supplemental Products
Reviews
Biological Activity
High affinity H3 receptor antagonist (Ki = 43.8 nM). Displays selectivity against H1 and H2 receptors (IC50 >10 μM). Increases the release of histamine in the cerebral cortex. Displays no activity at histamine methyltransferase in vitro at concentrations up to 3 μM. Brain penetrant.
High affinity H3 receptor antagonist (Ki = 43.8 nM). Displays selectivity against H1 and H2 receptors (IC50 >10 μM). Increases the release of histamine in the cerebral cortex. Displays no activity at histamine methyltransferase in vitro at concentrations up to 3 μM. Brain penetrant.
Technical Data
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M.Wt:317.47
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Formula:C19H31N3O
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Solubility:Soluble to 100 mM in DMSO and to 100 mM in ethanol
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Purity:>98
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Storage:Store at -20°C
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CAS No:152241-24-2
The technical data provided above is for guidance only.
For batch specific data refer to the Certificate of Analysis.
All Tocris products are intended for laboratory research use only.
Product Datasheets
VersaClone cDNA Plasmids
Description
Application
Cat#
Citations
Images
Human Histamine H3 R (NP_009163) VersaClone cDNA
RDC0344
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Mouse Histamine H3 R (NP_598610) VersaClone cDNA
RDC0728
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