GT 2016

Catalog # Availability Size / Price Qty
2419/10
2419/50
Cat.No. 2419 - GT 2016 | C19H31N3O | CAS No. 152241-24-2
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Description: Selective H3 antagonist

Chemical Name: 5-Cyclohexyl-1-[4-(1H-imidazol-5-yl)-1-piperidinyl]-1-pentanone

Purity: ≥98%

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Biological Activity

High affinity H3 receptor antagonist (Ki = 43.8 nM). Displays selectivity against H1 and H2 receptors (IC50 >10 μM). Increases the release of histamine in the cerebral cortex. Displays no activity at histamine methyltransferase in vitro at concentrations up to 3 μM. Brain penetrant.

Technical Data

M.Wt:
317.47
Formula:
C19H31N3O
Solubility:
Soluble to 100 mM in DMSO and to 100 mM in ethanol
Purity:
≥98%
Storage:
Store at -20°C
CAS No:
152241-24-2

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis. All Tocris products are intended for laboratory research use only.

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