Catalog Number: 5965
Chemical Name: 4-(2-Furanyl)-4,10-dihydro-2-methylpyrimido[1,2-a]benzimidazole-3-carboxylic acid-1-methylethyl ester
Biological Activity
High affinity A2B receptor antagonist (Ki = 3.49 nM). Exhibits >1000-fold selectivity for A2B over A1, A2A and A3 receptors.
Technical Data
  • M.Wt:
    337.37
  • Formula:
    C19H19N3O3
  • Solubility:
    Soluble to 20 mM in DMSO
  • Purity:
    >98%
  • Storage:
    Store at -20°C
  • CAS No:
    932191-62-3
The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis. All Tocris products are intended for laboratory research use only.
Background References
  1. Discovery of potent and highly selective A2B adenosine receptor antagonist chemotypes.
    El Maatougui et al.
    J.Med.Chem., 2016;59:1967
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