MA 2029

Catalog # Availability Size / Price Qty
4934/10
4934/50
Motilin Receptor Antagonists Small Molecule
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Description: Potent and selective, competitive motilin receptor antagonist; orally active

Chemical Name: 4-Fluoro-N-methyl-L-phenylalanyl-N-methyl-L-valyl-3-(1,1-dimethylethyl)-N-ethyl-L-tyrosinamide

Purity: ≥98%

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Biological Activity

Potent and selective, competitive motilin receptor antagonist (IC50 = 4.9 nM). Selective for the motilin receptor over a range of other receptors and ion channels. Inhibits motilin-induced duodenal muscle contractions in vitro. Also inhibits motilin-induced colonic and abdominal contractions in vivo. Orally active.

Technical Data

M.Wt:
556.71
Formula:
C31H45FN4O4
Solubility:
Soluble to 20 mM in 1eq. HCl and to 100 mM in DMSO
Purity:
≥98%
Storage:
Store at +4°C
CAS No:
287206-61-5

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
Tocris products are intended for laboratory research use only, unless stated otherwise.

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