Potent and competitive 5-HT6
= 7.2 nM, Ki
= 0.2 nM) that displays selectivity over other 5-HT and D2
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6-bicyclopiperazinyl-1-arylsulfonylindoles and 6-bicyclopiperidinyl-1-arylsulfonylindoles derivatives as novel, potent, and selective 5-HT6 receptor antagonists.
Isaac et al.