PNU 109291

2556 has been discontinued. View all 5-HT1D Receptor Agonists products.
  ( 1 citations )    
Product Datasheet
Catalog Number:2556
Chemical Name:(S)-3,4-Dihydro-1-[2-[4-(4-methoxyphenyl)-1-piperazinyl]ethyl]-N-methyl-1H-2-benzopyran-6-carboxamide
Product Details
Citations (1)
Reviews
Biological Activity
Potent and selective 5-HT1D receptor agonist that displays > 600-fold selectivity over 5-HT1A and 5-HT2A receptors and no activity at 5-HT1B, 5-HT1E, 5-HT2B, 5-HT2C, 5-HT6 and 5-HT7 receptors. Reduces dural plasma extravasation evoked by trigeminal ganglion stimulation.
Technical Data
  • M.Wt:
    409.52
  • Formula:
    C24H31N3O3
  • Solubility:
    Soluble to 100 mM in DMSO and to 100 mM in ethanol
  • Purity:
    >98
  • Storage:
    Store at +4°C
  • CAS No:
    187665-60-7
The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis. All Tocris products are intended for laboratory research use only.
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Citations:

The citations listed below are publications that use Tocris products. Selected citations for PNU 109291 include:

1 Citations: Showing 1 - 1

  1. 5-HT is a potent relaxant in rat superior mesenteric veins.
    Authors: Watts Et al.
    J Mol Neurosci  2015;3:e00103

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