Pristimerin

Catalog # Availability Size / Price Qty
3731/10
3731/50
Pristimerin | CAS No. 1258-84-0 | Monoacylglycerol Lipase Inhibitors
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Description: Potent, reversible MAGL inhibitor

Chemical Name: (9β,13α,14β,20α)-3-Hydroxy-9,13-dimethyl-2-oxo-24,25,26-trinoroleana-1(10),3,5,7-tetraen-29-oic acid methyl ester

Purity: ≥99%

Product Details
Citations (1)
Reviews

Biological Activity

Potent and reversible inhibitor of monoacylglycerol lipase (MGL) (IC50 = 93 nM). Also suppresses NF-κB activation via inhibition of proteasome chymotrypsin-like activity and IKKαβ. Displays antitumor, anti-inflammatory and antimicrobial activities.

Technical Data

M.Wt:
464.64
Formula:
C30H40O4
Solubility:
Soluble to 25 mM in DMSO and to 10 mM in ethanol
Purity:
≥99%
Storage:
Store at -20°C
CAS No:
1258-84-0

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
Tocris products are intended for laboratory research use only, unless stated otherwise.

Product Datasheets

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Citation for Pristimerin

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