Highly selective, water-soluble, human A2B
adenosine receptor antagonist. Ki
values are 53.4, > 10000 and > 10000 nM at human A2B
receptors respectively. Also selective versus rat A1
values are 2200 and 24000 nM respectively). Produces potent analgesic effects in vivo
The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
All Tocris products are intended for laboratory research use only.
Antinociceptive effects of novel A2B adenosine receptor antagonists.
Abo-Salem et al.
Preparation, properties, reactions, and adenosine receptor affinities of sulfophenylxanthine nitrophenyl esters: toward the development of sulfonic acid prodrugs with peroral bioavailability.
Yan and Muller
8-(Sulfostyryl)xanthines: water-soluble A2A-selective adenosine receptor antagonists.
Muller et al.
1,8-Disubstituted xanthine derivatives: synthesis of potent A2B-selective adenosine receptor antagonists.
Hayallah et al.
The citations listed below are publications that use Tocris products. Selected citations for PSB 1115 include:
Showing Results 1 - 9 of 9