Potent equilibrative nucleoside transporter 4 (ENT4) inhibitor (IC50
= 74.4 nM). Exhibits 20-fold and 80-fold selectivity for ENT4 over ENT2 and ENT1, respectively.
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All Tocris products are intended for laboratory research use only.
Dipyridamole analogs as pharmacological inhibitors of equilibrative nucleoside transporters. Identification of novel potent and selective inhibitors of the adenosine transporter function of human equilibrative nucleoside transporter 4 (hENT4).
Wang et al.