YIL 781

Catalog # Availability Size / Price Qty
3959/5
3959/25
Cat.No. 3959 - YIL 781 | C24H28FN3O2.HCl | CAS No. 875258-85-8
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Description: Ghrelin receptor (GHS-R1a) antagonist

Chemical Name: 6-(4-Fluorophenoxy)-2-methyl-3-[[(3S)-1-(1-methylethyl)-3-piperidinyl]methyl]-4(3H)-quinazolinone

Purity: ≥98%

Product Details
Citations (2)
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Biological Activity

Ghrelin receptor antagonist (GHS-R1a) (Ki = 17 nM). Displays no significant affinity for the motilin receptor (Ki = 6 μM). Blocks the effects of ghrelin on insulin secretion both in vivo and in vitro. Improves glucose homeostasis in vivo.

Technical Data

M.Wt:
445.96
Formula:
C24H28FN3O2.HCl
Solubility:
Soluble to 100 mM in DMSO and to 100 mM in water
Purity:
≥98%
Storage:
Desiccate at RT
CAS No:
875258-85-8

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis. All Tocris products are intended for laboratory research use only.

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Citations for YIL 781

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