5 results for "5-HT2C Receptor Antagonists Small Molecules and Peptides" in Products

5-HT2C Receptor Antagonists Small Molecules and Peptides

Serotonin 5-HT2C receptors, previously known as 5-HT1C receptors, are located primarily in the choroid plexus, cortex, limbic system and basal ganglia. 5-HT2C receptors play a role in CSF volume regulation, thermoregulation, penile erection and anxiety. The human 5-HT2C receptor gene has been localized to chromosome X (Xq24).

Dopamine antagonist with some D4 selectivity; also 5-HT2A/2C antagonist

Chemical Name: 8-Chloro-11-(4-methyl-1-piperazinyl)-5H-dibenzo[b,e][1,4]diazepine
Purity: ≥98%
Dopamine antagonist with some D4 selectivity; also 5-HT2A/2C antagonist
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Selective 5-HT2C antagonist

Chemical Name: 8-[5-(2,4-Dimethoxy-5-(4-trifluoromethylphenylsulphonamido)phenyl-5-oxopentyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione hydrochloride
Purity: ≥98%
Selective 5-HT2C antagonist
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Potent and selective 5-HT2B and 5-HT2C antagonist; orally active

Chemical Name: 3,5-Dihydro-5-methyl-N-3-pyridinylbenzo[1,2-b:4,5-b']dipyrrole-1(2H)-carboxamide hydrochloride
Purity: ≥98%
Potent and selective 5-HT2B and 5-HT2C antagonist; orally active
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Selective 5-HT2C antagonist; brain penetrant

Chemical Name: 6-Chloro-2,3-dihydro-5-methyl-N-[6-[(2-methyl-3-pyridinyl)oxy]-3-pyridinyl]-1H-indole-1-carboxyamide dihydrochloride
Purity: ≥98%
Selective 5-HT2C antagonist; brain penetrant
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5-HT2A and 5-HT2C antagonist; also D2-like partial agonist

Alternate Names: CU-32-085
Chemical Name: N'-[(8-α1,6-dimethylergolin-8-yl]-N,N-dimethylsulfamide hydrochloride
Purity: ≥98%
5-HT2A and 5-HT2C antagonist; also D2-like partial agonist
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