7 results for "Estrogen and Related Receptor Antagonists" in Products
Estrogen and Related Receptor Antagonists
Estrogen controls many cellular processes including growth, differentiation and function of the reproductive system. In females, estrogen's main targets are the ovaries, uterus, vagina and mammary glands. In the male, target organs are the testes, prostate and epididymis. Estrogen is also responsible for the growth and maintenance of the skeleton and the normal functioning of the cardiovascular and nervous systems.
Estrogen exerts most of its actions via estrogen receptors (ER). Estrogen ...
Estrogen receptor antagonist
| Alternate Names: | Fulvestrant |
| Chemical Name: | 7α,17β-[9-[(4,4,5,5,5-Pentafluoropentyl)sulfinyl]nonyl]estra-1,3,5(10)-triene-3,17-diol |
| Purity: | ≥98% |
High affinity and selective GPER antagonist
| Chemical Name: | (3aS*,4R*,9bR*)-4-(6-Bromo-1,3-benzodioxol-5-yl)-3a,4,5,9b-3H-cyclopenta[c]quinoline |
| Purity: | ≥98% |
Highly selective ERα antagonist
| Chemical Name: | 1,3-Bis(4-hydroxyphenyl)-4-methyl-5-[4-(2-piperidinylethoxy)phenol]-1H-pyrazole dihydrochloride |
| Purity: | ≥98% |
Selective ERβ antagonist
| Chemical Name: | 4-[2-Phenyl-5,7-bis(trifluoromethyl)pyrazolo[1,5-a]pyrimidin-3-yl]phenol |
| Purity: | ≥98% |
Selective GPER antagonist
| Chemical Name: | (±)-(3aR*,4S*,9bS*)-4-(6-Bromo-1,3-benzodioxol-5-yl)-3a,4,5,9b-tetrahydro-8-(1-methylethyl)-3H-cyclopenta[c]quinoline |
| Purity: | ≥98% |
ERα antagonist; also activates unfolded protein response; active in vivo
| Chemical Name: | 1,3-Dihydro-3,3-bis(4-hydroxyphenyl)-7-methyl-2H-indol-2-one |
| Purity: | ≥98% |
Potent and selective G protein-coupled estrogen receptor (GPER) antagonist
| Chemical Name: | N-[2-Cyclohexyl-4-(1-methylethyl)phenyl]-4-methoxybenzenemethanamine hydrochloride |
| Purity: | ≥98% |
