6 results for "Focal Adhesion Kinase Inhibitors" in Products

Focal Adhesion Kinase Inhibitors

Focal adhesion kinase (FAK), a non-receptor tyrosine kinase, is the first intracellular step in the signal transduction cascade initiated by the attachment of an integrin to the extracellular matrix at points known as focal adhesions. Therefore, FAK plays a key role in cellular migration and motility.

FAK has 3 functional domains: a focal adhesion targeting domain (FAT), a catalytic domain and a FERM domain, which mediates interactions with the cytoplasmic domains of integrins and growth ...

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Potent and selective FAK inhibitor

Chemical Name: 3,4-Dihydro-6-[[4-[[[3-(methylsulfonyl)phenyl]methyl]amino]-5-(trifluoromethyl)-2-pyrimidinyl]amino]-2(1H)-quinolinone
Purity: ≥98%
Potent and selective FAK inhibitor
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Selective FAK inhibitor

Alternate Names: Y15,NSC 677249
Chemical Name: 1,2,4,5-Benzenetetramine tetrahydrochloride
Selective FAK inhibitor
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Dual FAK/PYK2 inhibitor

Chemical Name: N-Methyl-N-[2-[[[2-[(2,3-dihydro-2-oxo-1H-indol-5-yl)amino]-5-(trifluoromethyl)-4-pyrimidinyl]amino]methyl]phenyl]methanesulfonamide
Purity: ≥98%
Dual FAK/PYK2 inhibitor
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Potent FAK inhibitor; orally bioavailable

Chemical Name: 2-[[2-[[2-Methoxy-4-(4-morpholinyl)phenyl]amino]-5-(trifluoromethyl)-4-pyridinyl]amino]-N-methylbenzamide
Purity: ≥98%
Potent FAK inhibitor; orally bioavailable
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Potent and selective FAK and Pyk2 inhibitor

Chemical Name: N-Methyl-4-[[4-[[[3-[methyl(methylsulfonyl)amino]-2-pyrazinyl]methyl]amino]-5-(trifluoromethyl)-2-pyrimidinyl]amino]benzamide
Purity: ≥98%
Potent and selective FAK and Pyk2 inhibitor
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Potent focal adhesion kinase (FAK) inhibitor

Chemical Name: 2-[[5-Chloro-2-[[3-methyl-1-(1-methylethyl)-1H-pyrazol-5-yl]amino]-4-pyridinyl]amino]-N-methoxybenzamide
Purity: ≥98%
Potent focal adhesion kinase (FAK) inhibitor
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