7 results for "GPR35" in Products

GPR35 Products

GPR35 is a rhodopsin-like G protein-coupled receptor (GPCR). GPR35 isoform B, also known as GPR35B, is longer at the N-terminus, compared to isoform A. Kynurenic acid, a tryptophan metabolite, and 2-acyl lysophosphatidic acid may act as endogenous ligands for GPR35. Human iNKT cells express GPR35 which is functionally active in reducing IL-4 releas...

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GPR35 agonist

Chemical Name: 2-(2-Propyloxyphenyl)-8-azapurin-6-one
Purity: ≥98%
GPR35 agonist
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Broad spectrum glutamatergic antagonist

Chemical Name: 4-Hydroxyquinoline-2-carboxylic acid
Purity: ≥98%
Broad spectrum glutamatergic antagonist
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GPR35 antagonist

Chemical Name: 1-(2,4-Difluorophenyl)-5-[[2-[[(1,1-dimethylehyl)amino]thioxomethyl]hydrazinylidene]methyl]-1H-pyrazole-4-carboxylic acid methyl ester
Purity: ≥98%
GPR35 antagonist
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GPR35 agonist

Chemical Name: 2-[3-Cyano-5-(3,4-dichlorophenyl)-4,5-dimethyl-2(5H)-furanylidene]propanedinitrile
Purity: ≥98%
GPR35 agonist
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GPR35 agonist; more potent than zaprinast (Cat. No. 0947)

Chemical Name: 4-[[2-[(2-Fluorophenyl)amino]-4-oxo-5(4H)-thiazolylidene]methyl]benzoic acid
Purity: ≥98%
GPR35 agonist; more potent than zaprinast (Cat. No. 0947)
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GPR35 antagonist

Chemical Name: 2-Hydroxy-4-[4-(5Z)-5-[(E)-2-methyl-3-phenylprop-2-enylidene]-4-oxo-2-sulfanylidene-1,3-thiazolidin-3-yl]butanoylamino]benzoic acid
Purity: ≥98%
GPR35 antagonist
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Na+/2Cl-/K+ (NKCC) symporter inhibitor

Chemical Name: 3-(Aminosulfonyl)-5-(butylamino)-4-phenoxybenzoic acid
Purity: ≥98%
Na+/2Cl-/K+ (NKCC) symporter inhibitor
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