5 results for "Nrf2" in Products

Nrf2 Products

NF-E2 related factor 2 (Nrf2) is a member of the cap 'n collar family of basic leucine zipper transcription factors. By binding antioxidant response elements (AREs), Nrf2 activates the transcription of genes encoding antioxidant and phase II drug-metabolizing enzymes needed to protect cells against oxidative damage. Transcriptional targets regulated by Nrf2 include genes encoding glutathione S-transferases, superoxide dismutase-1, and heme oxygenase-1.

Nrf2 signaling activator

Chemical Name: 1-(2-Cyano-3,12,28-trioxooleana-1,9(11)-dien-28-yl)-1H-imidazole
Purity: ≥98%
Nrf2 signaling activator
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Nrf2 activator; cell permeable

Chemical Name: 2-Methylenebutanedioic acid 4-octyl ester
Purity: ≥98%
Nrf2 activator; cell permeable
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Nrf2 activator

Chemical Name: N-[5-(2-Furanyl)-1,3,4-oxadiazol-2-yl]-N'-(2-pyridinylmethyl)urea
Purity: ≥98%
Nrf2 activator
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Nrf2 activator; inhibits Nrf2/Keap1 interaction

Chemical Name: (3S)-1-[4-[[(2,3,5,6-Tetramethylphenyl)sulfonyl]amino]-1-naphthalenyl]-3-pyrrolidinecarboxylic acid
Purity: ≥98%
Nrf2 activator; inhibits Nrf2/Keap1 interaction
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Inhibitor of Keap1- Nrf2 interaction

Alternate Names: LH601A
Chemical Name: (1S,2R)-2-[[(1S)-1-[(1,3-Dihydro-1,3-dioxo-2H-isoindol-2-yl)methyl]-3,4-dihydro-2(1H)-isoquinolinyl]carbonyl]cyclohexanecarboxylic acid
Purity: ≥98%
Inhibitor of Keap1- Nrf2 interaction
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