6 results for "PDE5A Small Molecules and Peptides" in Products

PDE5A Small Molecules and Peptides

PDE5A encodes a cGMP-binding, cGMP-specific phosphodiesterase, a member of the cyclic nucleotide phosphodiesterase family. This phosphodiesterase specifically hydrolyzes cGMP to 5'-GMP. It is involved in the regulation of intracellular concentrations of cyclic nucleotides and is important for smooth muscle relaxation in the cardiovascular system. Alternative splicing of this gene results in three transcript variants encoding distinct isoforms.

PDE inhibitor (non-selective)

Chemical Name: 3,7-Dihydro-1-methyl-3-(2-methylpropyl)-1H-purine-2,6-dione
Purity: ≥98%
PDE inhibitor (non-selective)
Loading...

GPR35 agonist

Chemical Name: 2-(2-Propyloxyphenyl)-8-azapurin-6-one
Purity: ≥98%
GPR35 agonist
Loading...

Adenosine transport inhibitor

Chemical Name: 2,6-bis(Diethanolamino)-4,8-dipiperidinopyrimido[5,4-d]pyrimidine
Purity: ≥98%
Adenosine transport inhibitor
Loading...

USP10 and USP13 inhibitor; inhibits autophagy

Chemical Name: 6-Fluoro-N-[(4-Fluorophenyl)methyl]-4-quinazolinamine
Purity: ≥98%
USP10 and USP13 inhibitor; inhibits autophagy
Loading...

Potent PDE5 inhibitor; orally active

Chemical Name: 1-[[3-(4,7-Dihydro-1-methyl-7-oxo-3-propyl-1H-pyrazolo[4,3-d]pyrimidin-5-yl)-4-ethoxyphenyl]sulfonyl]-4-methylpiperazine citrate
Purity: ≥98%
Potent PDE5 inhibitor; orally active
Loading...

Potent and highly selective PDE5 inhibitor; orally bioavailable

Alternate Names: GF196960
Chemical Name: (6R,12aR)-6-(1,3-Benzodioxol-5-yl)-2,3,6,7,12,12a-hexahydro-2-methylpyrazino[1',2':1,6]pyrido[3,4-b]indole-1,4-dione
Purity: ≥98%
Potent and highly selective PDE5 inhibitor; orally bioavailable
Loading...
Results Per Page
5 10 25 50
  • / 1