7 results for "V1a Vasopressin R/AVPR1A Small Molecules and Peptides" in Products
V1a Vasopressin R/AVPR1A Small Molecules and Peptides
AVPR1A acts as a receptor for arginine vasopressin and belongs to the subfamily of G protein-coupled receptors which includes AVPR1B, V2R and OXT receptors. Its activity is mediated by G proteins which stimulate a phosphatidylinositol-calcium second messenger system. AVPR1A mediates cell contraction and proliferation, platelet aggregation, release of coagulation factor and glycogenolysis. AVPR1A may be involved in social behaviors, including affiliation and attachment.
Antidiuretic hormone
| Alternate Names: | AVP |
| Purity: | ≥95% |
Selective, orally active vasopressin V1A receptor antagonist
| Alternate Names: | Relcovaptan |
| Chemical Name: | (2S)-1-[[(2R,3S)-5-Chloro-3-(2-chlorophenyl)-1-[(3,4-dimethoxyphenyl)sulfonyl]-2,3-dihydro-3-hydroxy-1H-indol-2-yl]carbonyl]-2-pyrrolidinecarboxamide |
| Purity: | ≥98% |
Selective vasopressin V1A antagonist
| Purity: | ≥95% |
Potent oxytocin receptor antagonist
| Purity: | ≥98% |
Orally active vasopressin V1 antagonist
| Chemical Name: | N-[3-[4-[[4-(3,4-Dihydro-2-oxo-1(2H)quinolinyl)-1-piperidinyl]carbonyl]phenoxy]propyl]-acetamide |
| Purity: | ≥98% |
Potent non-peptide oxytocin receptor partial agonist; also V1a receptor antagonist
| Chemical Name: | (2S)-N-[[4-[(4,10-Dihydro-1-methylpyrazolo[3,4-b][1,5]benzodiazepin-5(1H)-yl)carbonyl]-2-methylphenyl]methyl]-2-[(hexahydro-4-methyl-1H-1,4-diazepin-1-yl)thioxomethyl]-1-pyrrolidinecarboxamide |
| Purity: | ≥97% |
Potent and selective vasopressin V2 receptor antagonist; renoprotective and orally active
| Alternate Names: | OPC-41061 |
| Chemical Name: | N-[4-[(7-Chloro-2,3,4,5-tetrahydro-5-hydroxy-1H-1-benzazepin-1-yl)carbonyl]-3-methylphenyl]-2-methylbenzamide |
| Purity: | ≥98% |
