AC 4

   
Product Datasheet
Catalog Number:5464
Chemical Name:1,3,4,5-Tetrahydro-7,8-dihydro-N-[2-[4-[2-[4-(trifluoromethyl)phenyl]diazenyl]phenyl]ethyl]-2H-2-benzazepine-2-carbothioamide
Product Details
Supplemental Products
Reviews
Biological Activity
Photoswitchable TRPV1 channel blocker (IC50 = 3.1 μM). Acts as an antagonist in trans conformation during voltage gated activation. Also acts as an antagonist in the cis formation during capsaicin-induced TRPV1 currents. Switches conformation from cis to trans at 440 nm and trans to cis at 360 nm. Allows photoswitchable antagonist and an agonist to be applied at the same time.
Technical Data
  • M.Wt:
    514.56
  • Formula:
    C26H25F3N4O2S
  • Solubility:
    Soluble to 100 mM in DMSO and to 20 mM in water with gentle warming
  • Purity:
    >98
  • Storage:
    Store at -20°C
  • CAS No:
    1459809-09-6
The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis. All Tocris products are intended for laboratory research use only.
Product Datasheets

FAQs

No product specific FAQs exist for this product, however you may

View all Small Molecule FAQs
VersaClone cDNA Plasmids
Description Application Cat# Citations Images  

Rat Vanilloid R1/TRPV1 (NP_114188) VersaClone cDNA

RDC1967
View Sizes & Prices
Catalog# Size Price Stock Quantity
Loading Information....

Have you used AC 4?

Submit a review and receive a $25US/€18/£15/$25CAN amazon gift card if you include an image - $10US/€7/£6/$10CAN Amazon card for reviews without an image. Limited to verified customers in USA, Canada and Europe.

Tocris Bioscience is the leading supplier of novel and exclusive tools for life science research with over 30 years' experience in the industry. Tocris is a Bio-Techne brand.

Order Details

Contact Us to Order
reload

Feedback

Customer Information
Calculators

Molarity Calculator

Calculate the mass, volume, or concentration required for a solution.
=
x
x
g/mol

*When preparing stock solutions always use the batch-specific molecular weight of the product found on the vial label and SDS / CoA (available online).

R&D Systems Guarantee