AR-M 1000390 hydrochloride
Chemical Name: N,N-Diethyl-4-(phenyl-4-piperidinylidenemethyl)-benzamide hydrochloride
Biological ActivityAR-M 1000390 hydrochloride is a non-peptidic, low-internalizing δ-selective opioid receptor agonist; derivative of SNC 80 (Cat. No. 0764). Does not trigger acute desensitization of the analgesic response; reduces CFA-induced hyperalgesia. Brain penetrant following systemic administration.
The technical data provided above is for guidance only.
For batch specific data refer to the Certificate of Analysis.
Tocris products are intended for laboratory research use only, unless stated otherwise.
Pharmacological characterization of AR-M1000390 at human opioid delta receptors.
Marie et al.
Life Sci., 2003;73:1691
Ligand-directed trafficking of the δ-opioid receptor in vivo: Two paths toward analgesic tolerance.
Pradhan et al.
Citation for AR-M 1000390 hydrochloride
The citations listed below are publications that use Tocris products. Selected citations for AR-M 1000390 hydrochloride include:
1 Citation: Showing 1 - 1
A Genetically Encoded Biosensor Reveals Location Bias of Opioid Drug Action.
Authors: Stoeber Et al.
No product specific FAQs exist for this product, however you mayView all Small Molecule FAQs
VersaClone cDNA Plasmids
Reviews for AR-M 1000390 hydrochloride
There are currently no reviews for this product. Be the first to review AR-M 1000390 hydrochloride and earn rewards!
Have you used AR-M 1000390 hydrochloride?
Submit a review and receive an Amazon gift card.
$25/€18/£15/$25CAN/¥75 Yuan/¥1250 Yen for a review with an image
$10/€7/£6/$10 CAD/¥70 Yuan/¥1110 Yen for a review without an image