Catalog Number: 4335
Chemical Name: N,N-Diethyl-4-(phenyl-4-piperidinylidenemethyl)-benzamide hydrochloride
Biological Activity
Non-peptidic, low-internalizing δ-selective opioid receptor agonist; derivative of SNC 80 (Cat. No. 0764). Does not trigger acute desensitization of the analgesic response; reduces CFA-induced hyperalgesia. Brain penetrant following systemic administration.
Technical Data
  • M.Wt:
  • Formula:
  • Solubility:
    Soluble to 100 mM in water and to 100 mM in DMSO
  • Purity:
  • Storage:
    Store at -20°C
  • CAS No:
The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis. All Tocris products are intended for laboratory research use only.
Background References
  1. Pharmacological characterization of AR-M1000390 at human opioid delta receptors.
    Marie et al.
    Life Sci., 2003;73:1691
  2. Ligand-directed trafficking of the δ-opioid receptor in vivo: Two paths toward analgesic tolerance.
    Pradhan et al.
    J.Neurosci., 2010;30:16459
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