Estrogen receptor agonist. Also inhibits organic anion transporting polypeptide 1B1 (OATP1B1) (IC50
= 70 nM).
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All Tocris products are intended for laboratory research use only.
Estrogen regulation of the cytochrome P450 3A subfamily in humans.
Williams et al.
A cell-based high-throughput assay to identify inhibitors of organic anion transporting polypeptides 1B1 and 1B3.
Obaidat et al.
FASEB J., 2009;23:748