ISOX DUAL

Catalog # Availability Size / Price Qty
5806/10
5806/50
Cat.No. 5806 - ISOX DUAL | C31H41N5O3
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Description: Dual BRD4 and CBP/p300 bromodomain inhibitor

Chemical Name: [3-[4-[2-[5-(Dimethyl-1,2-oxazol-4-yl)-1-[2-(morpholin-4-yl)ethyl]-1H-1,3-benzodiazol-2-yl]ethyl]phenoxy]propyl]dimethylamine

Purity: ≥98%

Product Details
Reviews

Biological Activity

Dual CBP/p300 and BRD4 bromodomain inhibitor (IC50 values are 0.65 and 1.5 μM for CBP and BRD4 respectively). Downregulates IL-6, IL-1β and IFN-β in macrophages.

Technical Data

M.Wt:
531.69
Formula:
C31H41N5O3
Solubility:
Soluble to 100 mM in 1eq. HCl and to 50 mM in DMSO
Purity:
≥98%
Storage:
Store at +4°C

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis. All Tocris products are intended for laboratory research use only.

Additional Information

Licensing Caveats:
Sold for research purposes under agreement from Pfizer Inc.

Product Datasheets

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