U 99194 maleate
Chemical Name: 2,3-Dihydro-5,6-dimethoxy-N, N-dipropyl-1H-inden-2-amine maleate
Biological ActivityPotent, selective D3 antagonist. Ki values are 160, 2281 and > 10000 nM for human cloned D3, D2 and D4 receptors respectively.
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For batch specific data refer to the Certificate of Analysis.
Tocris products are intended for laboratory research use only, unless stated otherwise.
Heterogeneity of behavioural profile between three putative selective D3 DA receptor antagonists using an ethologically based approach.
Clifford and Waddington
A comparative in vitro and in vivo pharmacological characterization of the novel DA D3 receptor antagonists (+)-S 14297, nafadotride, GR 103,691 and U 99194.
Audinot et al.
DA D1 receptors synergize with D2, but not D3 or D4, receptors in the striatum without the involvement of action potentials.
LaHoste et al.
Citations for U 99194 maleate
The citations listed below are publications that use Tocris products. Selected citations for U 99194 maleate include:
2 Citations: Showing 1 - 2
Examining the Effects of Sodium Ions on the Binding of Antagonists to DA D 2 and D 3 Receptors
Authors: Newton Et al.
PLoS One 2016;11:e0158808
Prototypical antipsychotic drugs protect hippocampal neuronal cultures against cell death induced by growth medium deprivation.
Authors: Bastianetto Et al.
BMC Neurosci 2006;7:28
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