9 results for "Dopamine D2 R/DRD2" in Products
Dopamine D2 R/DRD2 Products
DRD2 encodes the D2 subtype of the dopamine receptor that inhibits adenylyl cyclase activity. Alternative splicing of this G protein-coupled receptor results in two transcript variants encoding different isoforms. DRD2 plays a major role in the neural circuitry that mediates behavioral control, an ability that is essential for adaptive responding and is compromised in a variety of common neuropsychiatric disorders.
Selective D2-like agonist
| Chemical Name: | (4aR-trans)-4,4a,5,6,7,8,8a,9-Octahydro-5-propyl-1H-pyrazolo[3,4-g]quinoline hydrochloride |
| Purity: | ≥98% |
High affinity D3 agonist (D3 ≥ D2 > D4)
| Chemical Name: | (4aR,10bR)-3,4a,4,10b-Tetrahydro-4-propyl-2H,5H-[1]benzopyrano-[4,3-b]-1,4-oxazin-9-ol hydrochloride |
| Purity: | ≥98% |
D2-like agonist (D2>D3>D4)
| Chemical Name: | (5'a)-2-Bromo-12'-hydroxy-2'-(1-methylethyl)-5'-(2-methylpropyl)ergotaman-3',6',18-trione mesylate |
| Purity: | ≥98% |
D2-like agonist (D2>D3>D4)
| Chemical Name: | N-[3-(Dimethylamino)propyl]-N-[(ethylamino)carbonyl]-6-(2-propenyl)ergoline-8-carboxamide |
| Purity: | ≥99% |
Selective D2 agonist
| Chemical Name: | (R)-5,6-Dihydro-5-(methylamino)-4H-imidazo[4,5,1-ij]quinolin-2(1H)-one (2Z)-2-butenedioate |
| Purity: | ≥98% |
Selective D2-like agonist
| Chemical Name: | 4-[2-(Dipropylamino)ethyl]-1,3-dihydro-2H-indol-2-one hydrochloride |
| Purity: | ≥98% |
D2 and D3 agonist
| Alternate Names: | N 0923 |
| Chemical Name: | (6S)-5,6,7,8-Tetrahydro-6-[propyl[2-(2-thienyl)ethyl]amino]-1-naphthalenol hydrochloride |
| Purity: | ≥99% |
High affinity D2 and 5-HT1A receptor partial agonist; also 5-HT2A antagonist
| Chemical Name: | 7-[4-[4-(2,3-Dichlorophenyl)-1-piperazinyl]butoxy]-3,4-dihydro-2(1H)-quinolinone |
| Purity: | ≥99% |
G protein-biased D2 partial agonist
| Chemical Name: | 5-Chloro-7-[[4-(2-pyridinyl)-1-piperazinyl]methyl]-8-quinolinol |
| Purity: | ≥98% |