50 results for "bromodomain-inhibitors&view=expanded" in Products

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(+)-JQ1

Catalog #: 4499
(2)
Citations (45)
Product Documents

Potent and selective BET bromodomain inhibitor; cell permeable

Chemical Name: (6S)-4-(4-Chlorophenyl)-2,3,9-trimethyl-6H-thieno[3,2-f][1,2,4]triazolo[4,3-a][1,4]diazepine-6-acetic acid 1,1-dimethylethyl ester
Purity: ≥98%
Potent and selective BET bromodomain inhibitor; cell permeable

PFI 1

Catalog #: 4445
Citations (5)
Product Documents

BET bromodomain inhibitor

Chemical Name: 2-Methoxy-N-(3-methyl-2-oxo-1,2,3,4-tetrahydroquinazolin-6-yl)benzenesulfonamide
Purity: ≥98%
BET bromodomain inhibitor

ent-LP 99

Catalog #: 5497
Product Documents

Negative Control for LP 99

Chemical Name: N-[(2S,3R)-2-(4-Chlorophenyl)-1-(1,2-dihydro-1,4-dimethyl-2-oxo-7-quinolinyl)-6-oxo-3-piperidinyl]-2-methyl-1-propanesulfonamide
Purity: ≥98%
Negative Control for LP 99

I-BET 151 dihydrochloride

Catalog #: 4650
(2)
Citations (10)
Product Documents

BET bromodomain inhibitor; also promotes differentiation of hiPSCs into megakaryocytes

Chemical Name: 7-(3,5-Dimethyl-4-isoxazolyl)-1,3-dihydroxy-8-methoxy-1-[(1R)-1-(2-pyridinyl)ethyl]-2H-imidazo[4,5-c]quinolin-2-one dihydrochloride
Purity: ≥98%
BET bromodomain inhibitor; also promotes differentiation of hiPSCs into megakaryocytes

GSK 9311 hydrochloride

Catalog #: 6203
Citations (1)
Product Documents

Negative control for GSK 6853

Chemical Name: N-[2,3-Dihydro-1,3-dimethyl-6-[(2R)-2-methyl-1-piperazinyl]-2-oxo-1H-benzimidazol-5-yl]-N-ethyl-2-methoxybenzamide hydrochloride
Purity: ≥98%
Negative control for GSK 6853

TP 238

Catalog #: 6670
Product Documents

CECR2 and BPTF/FALZ inhibitor

Chemical Name: N-[(3-(1H)-Pyrazol-1-yl)propyl)-6-(4-(3-(dimethylamino)propoxy)phenyl)-2-(methylsulfonyl)pyrimidin-4-amine hydrochloride
Purity: ≥98%
CECR2 and BPTF/FALZ inhibitor

MZ 1

Catalog #: 6154
Citations (19)
Product Documents

(+)-JQ1 based Degrader (PROTAC®) that preferentially degrades BRD4

Chemical Name: (2S,4R)-1-((S)-2-(tert-butyl)-17-((S)-4-(4-chlorophenyl)-2,3,9-trimethyl-6H-thieno[3,2-f][1,2,4]triazolo[4,3-a][1,4]diazepin-6-yl)-4,16-dioxo-6,9,12-trioxa-3,15-diazaheptadecanoyl)- 4-hydroxy-N-(4-(4-methylthiazol-5-yl)benzyl)pyrrolidine-2-carboxamide
Purity: ≥98%
Application of MZ 1 in HeLa Cells
(2)

I-BRD9

Catalog #: 5591
Citations (11)
Product Documents

Potent and selective BRD9 inhibitor

Chemical Name: 5-Ethyl-4,5-dihydro-4-oxo-N-(tetrahydro-1,1-dioxido-2H-thiopyran-4-yl)-7-[3-(trifluoromethyl)phenyl]thieno[3,2-c]pyridine-2-carboximidamide
Purity: ≥98%
Potent and selective BRD9 inhibitor

Bromosporine

Catalog #: 4758
Citations (2)
Product Documents

Broad spectrum bromodomain inhibitor

Chemical Name: N-[(6-3-Methanesulfonamido-4-methylphenyl)-3-methyl-[1,2,4]triazolo[4,3-b]pyridazin-8-yl]carbamate
Purity: ≥98%
Broad spectrum bromodomain inhibitor

SGC-CBP30

Catalog #: 4889
(1)
Citations (13)
Product Documents

Potent CBP/p300 BRD inhibitor

Chemical Name: 2-[2-(3-Chloro-4-methoxyphenyl)ethyl]-5-(dimethyl-1,2-oxazol-4-yl)-1-[(2S)-2-(morpholin-4-yl)propyl]-1H-1,3-benzodiazole
Purity: ≥98%
Potent CBP/p300 BRD inhibitor
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