8 results for "delta Opioid R/OPRD1 Small Molecules and Peptides" in Products
delta Opioid R/OPRD1 Small Molecules and Peptides
G protein-coupled receptors (GPCRs) are the largest family of membrane receptors that activate intracellular signaling cascades and undergo endocytosis, recycling, or degradation upon stimulation. The mu, delta and kappa opioid receptors are GPCRs of the nervous system, which control pain, stress, and addictive behaviors. The delta opioid receptor (DOR-1) is the stereo selective receptor for enkephalins and inhibits neurotransmitter release by reducing calcium ion currents and increasing potassium ion conductance.
Highly selective non-peptide δ agonist
| Chemical Name: | (+)-4-[(αR)-α-((2S,5R)-4-Allyl-2,5-dimethyl-1-piperazinyl)-3-methoxybenzyl]-N,N-diethylbenzamide |
| Purity: | ≥98% |
Selective δ agonist peptide
| Purity: | ≥95% |
δ selective peptide antagonist
| Purity: | ≥95% |
Selective, high affinity non-peptide δ1 agonist
| Alternate Names: | TAN 67 |
| Chemical Name: | (R*,S*)-(±)-2-Methyl-4aa-(3-hydroxyphenyl)-1,2,3,4,4a,5,12,12aa-octahydroquinolino[2,3,3-g]isoquinoline dihydrobromide |
| Purity: | ≥97% |
Selective δ agonist
| Alternate Names: | [D-Pen2,5]Enkephalin,[D-Pen2,D-Pen5]Enkephalin |
| Purity: | ≥95% |
Opioid receptor antagonist
| Chemical Name: | (5α)-17-(Cyclopropylmethyl)-4,5-epoxy-6-methylenemorphinan-3,14-diol hydrochloride |
| Purity: | ≥98% |
Potent positive allosteric modulator of δ receptors
| Chemical Name: | 3,4,5,6,7,9-Hexahydro-3,3,6,6-tetramethyl-9-[4-[(2-methylphenyl)methoxy]phenyl]-1H-xanthene-1,8(2H)-dione |
| Purity: | ≥98% |
Potent, selective non-peptide δ agonist
| Chemical Name: | 4-[(S)-[(2S,5R)-2,5-Dimethyl-4-(2-propenyl)-1-piperazinyl]phenylmethyl]-N,N-diethylbenzamide |
| Purity: | ≥98% |
