9 results for "Dopamine D2 R/DRD2" in Products

Dopamine D2 R/DRD2 Products

DRD2 encodes the D2 subtype of the dopamine receptor that inhibits adenylyl cyclase activity. Alternative splicing of this G protein-coupled receptor results in two transcript variants encoding different isoforms. DRD2 plays a major role in the neural circuitry that mediates behavioral control, an ability that is essential for adaptive responding and is compromised in a variety of common neuropsychiatric disorders.

Selective D2-like agonist

Chemical Name: (4aR-trans)-4,4a,5,6,7,8,8a,9-Octahydro-5-propyl-1H-pyrazolo[3,4-g]quinoline hydrochloride
Purity: ≥98%
Selective D2-like agonist
Loading...

High affinity D3 agonist (D3 ≥ D2 > D4)

Chemical Name: (4aR,10bR)-3,4a,4,10b-Tetrahydro-4-propyl-2H,5H-[1]benzopyrano-[4,3-b]-1,4-oxazin-9-ol hydrochloride
Purity: ≥98%
High affinity D3 agonist (D3 ≥ D2 > D4)
Loading...

D2-like agonist (D2>D3>D4)

Chemical Name: (5'a)-2-Bromo-12'-hydroxy-2'-(1-methylethyl)-5'-(2-methylpropyl)ergotaman-3',6',18-trione mesylate
Purity: ≥98%
D2-like agonist (D2>D3>D4)
Loading...

D2-like agonist (D2>D3>D4)

Chemical Name: N-[3-(Dimethylamino)propyl]-N-[(ethylamino)carbonyl]-6-(2-propenyl)ergoline-8-carboxamide
Purity: ≥99%
D2-like agonist (D2>D3>D4)
Loading...

Selective D2 agonist

Chemical Name: (R)-5,6-Dihydro-5-(methylamino)-4H-imidazo[4,5,1-ij]quinolin-2(1H)-one (2Z)-2-butenedioate
Purity: ≥98%
Selective D2 agonist
Loading...

Selective D2-like agonist

Chemical Name: 4-[2-(Dipropylamino)ethyl]-1,3-dihydro-2H-indol-2-one hydrochloride
Purity: ≥98%
Selective D2-like agonist
Loading...

D2 and D3 agonist

Alternate Names: N 0923
Chemical Name: (6S)-5,6,7,8-Tetrahydro-6-[propyl[2-(2-thienyl)ethyl]amino]-1-naphthalenol hydrochloride
Purity: ≥99%
D2 and D3 agonist
Loading...

High affinity D2 and 5-HT1A receptor partial agonist; also 5-HT2A antagonist

Chemical Name: 7-[4-[4-(2,3-Dichlorophenyl)-1-piperazinyl]butoxy]-3,4-dihydro-2(1H)-quinolinone
Purity: ≥99%
High affinity D2 and 5-HT1A receptor partial agonist; also 5-HT2A antagonist
Loading...

G protein-biased D2 partial agonist

Chemical Name: 5-Chloro-7-[[4-(2-pyridinyl)-1-piperazinyl]methyl]-8-quinolinol
Purity: ≥98%
G protein-biased D2 partial agonist
Loading...
Results Per Page
5 10 25 50
  • / 1