8 results for "FGF Receptor Inhibitors" in Products

FGF Receptor Inhibitors

Fibroblast growth factors (FGFs) (FGF1 - 10 and 16 - 23) are mitogenic signaling molecules that have roles in angiogenesis, wound healing, cell migration, neural outgrowth and embryonic development. FGFs bind heparan sulfate glycosaminoglycans (HSGAGs), which facilitates dimerization (activation) of FGF receptors (FGFRs).

FGFRs are transmembrane catalytic receptors that have intracellular tyrosine kinase activity. There are four human genes encoding FGFRs, which produce seven different receptors ...

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Potent FGFR and VEGFR inhibitor

Alternate Names: PF-02969207,PNU-0290908
Chemical Name: 2-[(1,2-Dihydro-2-oxo-3H-indol-3-ylidene)methyl]-4-methyl-1H-pyrrole-3-propanoic acid
Purity: ≥95%
Potent FGFR and VEGFR inhibitor
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FGFR1 and -3 inhibitor

Chemical Name: N-[2-[[4-(Diethylamino)butyl]amino]-6-(3,5-dimethoxyphenyl)pyrido[2,3-d]pyrimidin-7-yl]-N'-(1,1-dimethylethyl)urea
Purity: ≥98%
FGFR1 and -3 inhibitor
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Potent VEGFR, PDGFR and FGFR inhibitor

Chemical Name: Methyl (Z)-3-[[[4-(N-methyl-2-(4-methylpiperazin-1-yl)acetamido)phenyl)amino)(phenyl)methylene]-2-oxoindoline-6-carboxylate
Purity: ≥98%
Potent VEGFR, PDGFR and FGFR inhibitor
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Potent Src inhibitor; also inhibits FGFR1, PDGFRβ and Wee1

Chemical Name: 6-(2,6-Dichlorophenyl)-2-[[4-[2-(diethylamino)ethoxy]phenyl]amino]-8-methylpyrido[2,3-d]pyrimidin-7(8H)-one dihydrochloride
Purity: ≥98%
Potent Src inhibitor; also inhibits FGFR1, PDGFRβ and Wee1
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Selective FGFR inhibitor

Chemical Name: N-[6-(2,6-Dichlorophenyl)-2-[[4-(diethylamino)butyl]amino]pyrido[2,3-d]pyrimidin-7-yl]-N'-(1,1-dimethylethyl)urea
Purity: ≥97%
Selective FGFR inhibitor
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Potent multi-kinase and pan-Bcr-Abl inhibitor

Alternate Names: Ponatinib
Chemical Name: 3-(2-Imidazo[1,2-b]pyridazin-3-ylethynyl)-4-methyl-N-[4-[(4-methyl-1-piperazinyl)methyl]-3-(trifluoromethyl)phenyl]-benzamide
Purity: ≥98%
Potent multi-kinase and pan-Bcr-Abl inhibitor
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Potent inhibitor of VEGFR, PDGFR and FGFR

Chemical Name: 4-[(4-Fluoro-2-methyl-1H-indol-5-yl)oxy]-6-methoxy-7-[3-(1-pyrrolidinyl)propoxy]quinazoline
Purity: ≥98%
Potent inhibitor of VEGFR, PDGFR and FGFR
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Potent and selective FGFR inhibitor

Chemical Name: rel-N-[5-[2-(3,5-Dimethoxyphenyl)ethyl]-1H-pyrazol-3-yl]-4-[(3R,5S)-3,5-dimethyl-1-piperazinyl]benzamide
Purity: ≥98%
Potent and selective FGFR inhibitor
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