12 results for "CaM Kinase Inhibitors" in Products

CaM Kinase Inhibitors

CaM kinase II inhibitor; also K+ channel blocker (KV)

Chemical Name: N-[2-[[[3-(4-Chlorophenyl)-2-propenyl]methylamino]methyl]phenyl]-N-(2-hydroxyethyl)-4-methoxybenzenesulphonamide
Purity: ≥98%
CaM kinase II inhibitor; also K+ channel blocker (KV)
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Selective CaM kinase kinase inhibitor

Chemical Name: 7-Oxo-7H-benzimidazo[2,1-a]benz[de]isoquinoline-3-carboxylic acid acetate
Purity: ≥98%
Selective CaM kinase kinase inhibitor
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Non-competitive P2X7 antagonist

Chemical Name: 4-[(2S)-2-[(5-isoquinolinylsulfonyl)methylamino]-3-oxo-3-(4-phenyl-1-piperazinyl)propyl] phenyl isoquinolinesulfonic acid ester
Purity: ≥98%
Non-competitive P2X7 antagonist
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CaM kinase II inhibitor; water soluble version of KN 93 (Cat. No. 1278)

Chemical Name: N-[2-[[[3-(4-Chlorophenyl)-2-propenyl]methylamino]methyl]phenyl]-N-(2-hydroxyethyl)-4-methoxybenzenesulphonamide phosphate
Purity: ≥98%
CaM kinase II inhibitor; water soluble version of KN 93 (Cat. No. 1278)
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Selective CaM kinase II inhibitor

Alternate Names: AIP
Purity: ≥95%
Selective CaM kinase II inhibitor
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CaM kinase III (eEF-2 kinase) inhibitor

Chemical Name: 1-Hexadecyl-2-methyl-3-(phenylmethyl)-1H-imidazolium iodide
CaM kinase III (eEF-2 kinase) inhibitor
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CaM kinase II inhibitor; enhanced cell permeable derivative of Autocamtide-2-related inhibitory peptide

Alternate Names: Myr-AIP,AIP Myristoylated
Purity: ≥95%
CaM kinase II inhibitor; enhanced cell permeable derivative of Autocamtide-2-related inhibitory peptide
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Potent CaM kinase I inhibitor

Chemical Name: 2-[(3S)-3-Amino-1-piperidinyl]-4-[[2,6-bis(1-methylethyl)-4-pyridinyl]amino]-5-pyrimidinecarboxamide
Purity: ≥98%
Potent CaM kinase I inhibitor
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Potent and selective calcium/calmodulin-dependent serine protein kinase (CASK) inhibitor

Chemical Name: 4-(Cyclopentylamino)-2-((2,5-dibromo-4-methylbenzyl)amino)-N-(3-(2-oxooxazolidin-3-yl)propyl)pyrimidine-5-carboxamide
Purity: ≥98%
Potent and selective calcium/calmodulin-dependent serine protein kinase (CASK) inhibitor
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Potent and selective CAMKK1/2 inhibitor

Chemical Name: 2-Cyclopentyl-4-[5-(3-methylphenyl)furo[2,3-b]pyridin-3-yl]benzoic acid
Purity: ≥95%
Potent and selective CAMKK1/2 inhibitor
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Staurosporine synthesized to Ancillary Material Grade

Chemical Name: [9S-(9α,10β,11β,13α)]-2,3,10,11,12,13-Hexahydro-10-methoxy-9-methyl-11-(methylamino)-9,13-epoxy-1H,9H-diindolo[1,2,3-gh:3',2',1'-lm]pyrrolo[3,4-j][1,7]benzodiazonin-1-one
Purity: ≥98%
Staurosporine synthesized to Ancillary Material Grade
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CaM kinase III (eEF-2 kinase) inhibitor

Chemical Name: 7-Amino-1-cyclopropyl-3-ethyl-1,2,3,4-tetrahydro-2,4-dioxopyrido[2,3-d]pyrimidine-6-carboxamide
Purity: ≥98%
CaM kinase III (eEF-2 kinase) inhibitor
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