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Peripherally acting μ agonist; Ca2+ channel blocker
α1 antagonist, L-type Ca2+ channel blocker
α1 antagonist, L-type Ca2+ channel blocker. Less active enantiomer of Niguldipine hydrochloride (Cat. No. 1123)
Dual CaV1.x and CaV2.x blocker
CaV1.x blocker; (R)-(+)-enantiomer of (±)-Bay K 8644; also TMEM176B inhibitor
Allosteric Calcium-sensing receptor (CaSR) agonist; also CYP2D2 inhibitor and Ca2+ channel blocker; orally bioavailable
Inhibits KRas localization to the plasma membrane; also L-type calcium channel blocker