12 results for "ER alpha/NR3A1 Small Molecules and Peptides" in Products
ER alpha/NR3A1 Small Molecules and Peptides
Estrogen receptor alpha (ER alpha, NR3A1) is a member of the steroid receptor family. The natural ligand for ER is the classic estrogenic compound 17 beta-estradiol. ER alpha is expressed in a wide variety of tissues such as bones, uterus, bladder, ovary, prostate, testis, epididymis, kidney, breast, heart, vessel wall, pituitary and hypothalamus. ...
Estrogen receptor antagonist
| Alternate Names: | Fulvestrant |
| Chemical Name: | 7α,17β-[9-[(4,4,5,5,5-Pentafluoropentyl)sulfinyl]nonyl]estra-1,3,5(10)-triene-3,17-diol |
| Purity: | ≥98% |
Metabolite of tamoxifen (Cat. No. 0999)
| Alternate Names: | 4-OH-TAM |
| Chemical Name: | 4-[(1Z)-1-[4-[2-(Dimethylamino)ethoxy]phenyl]-2-phenyl-1-buten-1-yl]phenol |
| Purity: | ≥98% |
Estrogen receptor partial agonist/antagonist
| Chemical Name: | (Z)-2-[4-(1,2-Diphenyl-1-butenyl)phenoxy]-N,N-dimethylethanamine citrate |
| Purity: | ≥98% |
Highly selective ERα antagonist
| Chemical Name: | 1,3-Bis(4-hydroxyphenyl)-4-methyl-5-[4-(2-piperidinylethoxy)phenol]-1H-pyrazole dihydrochloride |
| Purity: | ≥98% |
Estrogen receptor partial agonist/antagonist
| Chemical Name: | 2-[4-[(1Z)-1,2-Diphenyl-1-buten-1-yl]phenoxy]-N,N-dimethylethanamine |
| Purity: | ≥98% |
Potent and selective ERα Degrader (SNIPER)
| Chemical Name: | (2S)-N-[(1S)-1-Cyclohexyl-2-[(2S)-2-[4-[3-[[14-[4-[1-(4-hydroxyphenyl)-2-phenyl-1-buten-1-yl]phenoxy]-12-methyl-11-oxo-3,6,9-trioxa-12-azatetradec-1-yl]oxy]benzoyl]-2-thiazolyl]-1-pyrrolidinyl]-2-oxoethyl]-2-(methylamino)propanamide |
| Purity: | ≥98% |
EGFR kinase inhibitor. Also estrogen and PPARγ ligand
| Chemical Name: | 5,7-Dihydroxy-3-(4-hydroxyphenyl)-4H-1-benzopyran-4-one |
| Purity: | ≥98% |
Selective estrogen receptor modulator (SERM)
| Alternate Names: | LY 139481,Keoxifene |
| Chemical Name: | [6-Hydroxy-2-(4-hydroxyphenyl)benzo[b]thien-3-yl][4-[2-(1-piperidinyl)ethoxy]phenyl]-methanone hydrochloride |
| Purity: | ≥98% |
Subtype-selective ERα agonist
| Chemical Name: | 4,4',4''-(4-Propyl-[1H]-pyrazole-1,3,5-triyl)trisphenol |
| Purity: | ≥98% |
Potent subtype-selective ligand; ERα agonist/ERβ antagonist
| Chemical Name: | (R,R)-5,11-Diethyl-5,6,11,12-tetrahydro-2,8-chrysenediol |
| Purity: | ≥98% |
ERα antagonist; also activates unfolded protein response; active in vivo
| Chemical Name: | 1,3-Dihydro-3,3-bis(4-hydroxyphenyl)-7-methyl-2H-indol-2-one |
| Purity: | ≥98% |
Selective estrogen receptor modulator (SERM), selective for ERα
| Chemical Name: | [6-Hydroxy-2-(4-hydroxyphenyl)benzo[b]thien-3-yl]-[4-[4-(1-methylethyl)-1-piperazinyl]phenyl]methanone |
| Purity: | ≥98% |
