10 results for "HIF Inhibitors" in Products

HIF Inhibitors

HIF-1α inhibitor; down-regulates HIF-1α protein synthesis

Chemical Name: N,N'-(Dithiodi-2,1-ethanediyl)bis[2,5-dichlorobenzenesulfonamide
Purity: ≥98%
HIF-1α inhibitor; down-regulates HIF-1α protein synthesis
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Thioredoxin-1 inhibitor

Alternate Names: IV-2
Chemical Name: 2-[(1-Methylpropyl)dithio]-1H-imidazole
Purity: ≥98%
Thioredoxin-1 inhibitor
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Prolyl hydroxylase inhibitor

Chemical Name: N-(2-Methoxy-2-oxoacetyl)glycine methyl ester
Purity: ≥97%
Prolyl hydroxylase inhibitor
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Highly potent and selective HIF-1α inhibitor

Alternate Names: Quinomycin A
Chemical Name: N-(2-Quinoxalinylcarbonyl)-O-[N-(2-quinoxalinylcarbonyl)-D-seryl-L-alanyl-3-mercapto-N,S-dimethylcysteinyl-N-methyl-L-valyl]-D-seryl-L-alanyl-N-methylcysteinyl-N-methyl-L-valine-(81)-lactone-cyclic (37)-thioether
Purity: ≥98%
Highly potent and selective HIF-1α inhibitor
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Malate dehydrogenase-2 (MDH2) inhibitor; also inhibits HIF-1α

Alternate Names: CAY 10585
Chemical Name: Methyl 4-hydroxy-3-[[2-(4-tricyclo[3.3.1.13,7]dec-1-ylphenoxy)acetyl]amino]benzoate
Purity: ≥98%
Malate dehydrogenase-2 (MDH2) inhibitor; also inhibits HIF-1α
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High affinity and selective HIF-2α inhibitor

Chemical Name: N-(3-Chloro-5-fluorophenyl)-4-nitro-2,1,3-benzoxadiazol-5-amine
Purity: ≥98%
High affinity and selective HIF-2α inhibitor
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Potent HIF-1α inhibitor

Chemical Name: N-(2,3-Dihydro-1,4-benzodioxin-6-yl)-1,4-dihydroindeno[1,2-c]pyrazol-3-amine
Purity: ≥98%
Potent HIF-1α inhibitor
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HIF α-subunit inhibitor

Chemical Name: 2-Oxo-2-(p-tolyl)ethyl 3-(2,4-dinitrobenzamido)benzoate
Purity: ≥98%
HIF α-subunit inhibitor
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Potent, selective HIF-1α prolyl hydroxylase-2 (PHD2) inhibitor

Chemical Name: N-[[1,2-Dihydro-4-hydroxy-2-oxo-1-(phenylmethyl)-3-quinolinyl]carbonyl]glycine
Purity: ≥98%
Potent, selective HIF-1α prolyl hydroxylase-2 (PHD2) inhibitor
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HIF-prolyl hydroxylase-2 (PHD2) inhibitor; antioxidant

Chemical Name: 7-[(4-Chlorophenyl)[(3-hydroxy-2-pyridinyl)amino]methyl]-8-quinolinol
Purity: ≥97%
HIF-prolyl hydroxylase-2 (PHD2) inhibitor; antioxidant
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